Affinity DataKi: 82.5nMAssay Description:Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assayMore data for this Ligand-Target Pair
Affinity DataKi: 83nMAssay Description:Opioid receptor delta 1 binding affinity by displacement of radioligand [3H][D-Pen]-enkephalin (DPDPE) from rat brain membrane synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Binding affinity against Opioid receptor delta 1 in P2 membrane preparation of rat brain by [3H]DADLE displacement.More data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 179nMAssay Description:Displacement of [3H]deltorphin II from rat delta opioid receptor in brain P2 synaptosomesMore data for this Ligand-Target Pair
Affinity DataKi: 192nMAssay Description:Binding affinity of the compound against Opioid receptor delta 1 using [3H]-DT in rat brain synaptosomes was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 295nMAssay Description:Inhibition of [3H]-naloxone binding to rat brain homogenate Opioid receptor deltaMore data for this Ligand-Target Pair
Affinity DataKi: 929nMAssay Description:Binding affinity to DOP (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]-NLT from Opioid receptor delta 1 of adult male mouse brain.More data for this Ligand-Target Pair
Affinity DataIC50: 15.2nMAssay Description:Functional bioactivity against delta opioid receptor in mouse vas deferensMore data for this Ligand-Target Pair
Affinity DataIC50: 16.5nMAssay Description:In vitro inhibitory activity against electrically evoked contractions of in mouse vas deferens (MVD)More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Agonist activity at delta-type opioid receptor in mouse vas deferens assessed as inhibition of electrically stimulated contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:In vitro opioid receptor delta mediated mouse vas deferens (MVD) assayMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:In vitro biological activity by electrically induced smooth muscle contractions in mouse vas deferens (Opioid receptor delta 1); inhibitory concentra...More data for this Ligand-Target Pair
Affinity DataIC50: 74nMAssay Description:Antagonist activity at mouse brain homogenate DOPMore data for this Ligand-Target Pair
Affinity DataIC50: 197nMAssay Description:Displacement of [3H]DPDPE from delta opioid receptor expressed in CHO cells after 90 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 210nMAssay Description:Evaluated for the inhibition of [3H]DADLE binding to Opioid receptor delta 1 of guinea pig brainMore data for this Ligand-Target Pair
Affinity DataIC50: 294nMAssay Description:Displacement of [3H]DSLET from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Evaluated for its affinity towards Opioid receptor delta 1 in rat fore brain by displacing the radioligand [3H]-DPDPE.More data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Binding affinity to delta-type opioid receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 295nMAssay Description:Agonist activity at delta-type opioid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 320nMAssay Description:Displacement of [3H]- DPDPE from delta opioid receptor in rat brain membraneMore data for this Ligand-Target Pair