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Found 3 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM50050516'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Trustees Of Tufts College

US Patent
LigandPNGBDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50:  1.30nMAssay Description:This assay is described in Bachovchin et al. Nature Chemical Biology 10, 656-663 (2014). Briefly, purified enzymes are coupled to Luminex microsphere...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Trustees Of Tufts College

US Patent
LigandPNGBDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50:  95nMAssay Description:In vitro for inhibition of Dipeptidylpeptidase IV.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Trustees Of Tufts College

US Patent
LigandPNGBDBM50050516(Boronic acid derivative | CHEMBL63726 | US11096924...)
Affinity DataIC50:  1.30E+3nMAssay Description:EnzymesRecombinant human DPPIV (R&D Systems, Cat. No. 1180-SE)Recombinant human DPP8 (Enzo Life Sciences, Cat. No. BML-SE527)Recombinant human DPP9 (...More data for this Ligand-Target Pair
In DepthDetails US Patent