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Found 3 Enz. Inhib. hit(s) with Target = 'Epidermal growth factor receptor' and Ligand = 'BDBM318899'
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Neupharma

US Patent
LigandPNGBDBM318899(N-(3-(2-((4-(2-methoxyethoxy)phenyl)amino)quinazol...)
Affinity DataIC50: >500nMAssay Description:The compound of Formula I binds to a kinase selected from the group consisting of EGFR, EGFR L858R, EGFR T790M, EGFR del E746-A750, or EGFR L858R/T79...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Neupharma

US Patent
LigandPNGBDBM318899(N-(3-(2-((4-(2-methoxyethoxy)phenyl)amino)quinazol...)
Affinity DataIC50: >500nMAssay Description:EGFR: The 2×EGFR (ErbB1)/Tyr 04 mixture is prepared in 50 mM HEPES pH 7.5, 0.01% BRIJ-35, 10 mM MgCl2, 4 mM MnCl2, 1 mM EGTA, 2 mM DTT. The final 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Neupharma

US Patent
LigandPNGBDBM318899(N-(3-(2-((4-(2-methoxyethoxy)phenyl)amino)quinazol...)
Affinity DataIC50: >500nMAssay Description:(i) Peptide/Kinase Mixtures for measurement of EGFR (ErbB1):The 2×EGFR (ErbB1)/Tyr 04 mixture is prepared in 50 mM HEPES pH 7.5, 0.01% BRIJ-35, 10 mM...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent