Found 35 Enz. Inhib. hit(s) with Target = 'Estrogen receptor' and Ligand = 'BDBM20607' 
Affinity DataKi: 31.2nMAssay Description:Displacement of [2,4,6,7-3H]estradiol from human ERalpha expressed in HeLa cells after 18 hrs by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 1.5nMAssay Description:Inhibition of estrogen receptor-alpha (unknown origin) by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Displacement of [3H]-E2 from human ER-alpha incubated for 16 to 20 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 8.40nMAssay Description:Displacement of radioligand from Estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Binding affinity to ERalpha receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Antagonist activity at Gal4 DBD-fused human ERalpha LBD expressed in HEK293T cells assessed as inhibition of estradiol-induced transcriptional activa...More data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Displacement of [3H]-17-beta-estradiol from human estrogen receptor alphaMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Antagonist activity at estrogen receptor in human T47D cells incubated for 18 hrs by ultra high sensitivity luminescence reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Binding affinity to human ERalphaMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Displacement of fluorescein-labeled estradiol (fluoromone) from human recombinant full-length untagged estrogen receptor alpha expressed in Spodopter...More data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Displacement of fluorescein-labeled estrogen from human recombinant ERalpha by fluorescence polarization based competitive binding affinity assayMore data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Antagonist activity at ERalpha (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 69nMAssay Description:Displacement of fluorescent labeled-ligand from ERalpha (unknown origin) by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of fluorescein labeled estradiol from human recombinant ERalpha expressed in baculovirus infected insect cells by fluorescence polarizat...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of fluorescent estrogen ligand from recombinant human full length untagged ERalpha expressed in baculovirus infected insect cells incuba...More data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of fluorescein-labeled estradiol (fluoromone) from human recombinant full-length estrogen receptor alpha after 2 hrs by fluorescence pol...More data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:Displacement of [3H]E2 from human recombinant ERalpha assessed as receptor binding after 45 mins by scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 222nMAssay Description:Inhibition of estrogen receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 222nMAssay Description:Displacement of Fluormone ES2 Green from human recombinant full length ERalpha expressed in insect cells measured up to 4 hrs by fluorescence polariz...More data for this Ligand-Target Pair
Affinity DataIC50: 226nMAssay Description:Displacement of [3H]E2 from GST-fused ERalpha-LBD (unknown origin) expressed in Escherichia coli BL21 incubated for 1 hr by liquid scintillation coun...More data for this Ligand-Target Pair
Affinity DataIC50: 341nMAssay Description:Antagonist activity at full length ERalpha (unknown origin) expressed in human HeLa cells incubated for 24 hrs by ERE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Antiestrogenic activity in MCF-7-2a cells as concentration required to reduce estradiol effect by 50%More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of fluorescein-labeled estrogen ligand from recombinant ER-alpha (unknown origin) incubated for 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.42E+3nMAssay Description:Displacement of Fluormone ES2 Green from full length human ER-alpha expressed in insect cells after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+3nMAssay Description:Displacement of fluorescent estrogen ligand from recombinant human full length untagged ERalpha expressed in Spodoptera frugiperda insect cells measu...More data for this Ligand-Target Pair
Affinity DataIC50: 1.61E+3nMAssay Description:Antagonist activity at ERalpha in human MCF7 cells assessed as inhibition of estrogen-induced transcription preincubated overnight followed by estrog...More data for this Ligand-Target Pair
Affinity DataIC50: 1.61E+3nMAssay Description:Induction of selective estrogen receptor alpha degradation in human MCF7 cells harboring TK-ERE-Luc assessed as reduction in estradiol-induced transc...More data for this Ligand-Target Pair
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human full-length ERalpha expressed in non-human mammalian expression system assessed as inhibition of 17beta-estradiol-induce...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:Antagonist activity at ERalpha receptor LBD expressed in yeast AH109 cells assessed as inhibition of interaction with SRC1 after 24 hrs by alpha-gala...More data for this Ligand-Target Pair
Affinity DataIC50: 2.54E+3nMAssay Description:Antagonist activity at ERalpha expressed in yeast assessed as inhibition of E2-induced alpha-galactosidase activityMore data for this Ligand-Target Pair
Affinity DataIC50: 2.67E+3nMAssay Description:Displacement of fluorescent estrogen ligand from recombinant human ERalpha expressed in insect cells incubated for 2 hrs by polarizationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at ERalpha receptor in human MCF7 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.54E+3nMAssay Description:Antagonist activity at human estrogen receptor-alpha by yeast two-hybrid assay in presence of SRC1More data for this Ligand-Target Pair
Affinity DataEC50: 622nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assay was performed by using 96-well microtiterplates containing ER, 17beta-estradiol, and the test compound to be tested and SPA...More data for this Ligand-Target Pair
Affinity DataEC50: 622nMpH: 7.4 T: 2°CAssay Description:Radioligand binding assay was performed by using 96-well microtiterplates containing ER, 17beta-estradiol, and the test compound to be tested and SPA...More data for this Ligand-Target Pair
