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Found 2 Enz. Inhib. hit(s) with Target = 'Free fatty acid receptor 1' and Ligand = 'BDBM294015'
TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM294015(5-((2S)-2-(4-((3-(4-(2- Methoxyethoxy)-2- methylph...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human GPR40 assessed as increase in intracellular calcium flux by cell based FLIPR assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFree fatty acid receptor 1(Homo sapiens (Human))TBA
LigandPNGBDBM294015(5-((2S)-2-(4-((3-(4-(2- Methoxyethoxy)-2- methylph...)
Affinity DataEC50:  13nMT: 2°CAssay Description:Compounds were tested in a calcium flux assay using transfected HEK293 cells stably expressing either human GPR40 or rat GPR40. Human GPR40 expressin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent