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Found 2 Enz. Inhib. hit(s) with Target = 'G-protein coupled bile acid receptor 1' and Ligand = 'BDBM398271'
TargetG-protein coupled bile acid receptor 1(Mus musculus)
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  17nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetG-protein coupled bile acid receptor 1(Homo sapiens (Human))
Universite De Lille 2 Droit Et Sante

US Patent
LigandPNGBDBM398271(US10323016, Example 8)
Affinity DataEC50:  260nMAssay Description:In the following tables TGR5 activation by compounds and subsequent increase in intracellular cAMP were evaluated using a luciferase reporter gene as...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent