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Found 2 Enz. Inhib. hit(s) with Target = 'Gamma-butyrobetaine dioxygenase' and Ligand = 'BDBM50008027'
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research And Study Centre

Curated by ChEMBL
LigandPNGBDBM50008027(CHEMBL3234384)
Affinity DataIC50:  90nMAssay Description:Inhibition of human recombinant BBOX expressed in Saccharomyces cerevisiae AH22 assessed as formation of carnitine from gamma-butyrobetaine preincuba...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGamma-butyrobetaine dioxygenase(Homo sapiens (Human))
Latvian Biomedical Research And Study Centre

Curated by ChEMBL
LigandPNGBDBM50008027(CHEMBL3234384)
Affinity DataKd:  9.30E+3nMAssay Description:Binding affinity to purified human BBOX by isothermal titration calorimetry analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed