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Found 2 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Ligand = 'BDBM50119557'
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50119557(CHEMBL3617575)
Affinity DataKi:  20nMAssay Description:Displacement of [125I]-glucagon from full length human glucagon receptor expressed in HEK293 cell membranes after 2 hrs by scintillation counting ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50119557(CHEMBL3617575)
Affinity DataIC50:  4nMAssay Description:Antagonist activity at human glucagon receptor expressed in HEK293 cell membranes assessed as inhibition of glucagon-stimulated intracellular cAMP fo...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed