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Found 3 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50197425'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197425(CHEMBL440227 | [4-({[4-((9S,11R,13S,14S,17S)-17-hy...)
Affinity DataKi:  1.80nMAssay Description:Displacement of radiolabeled Dexamethasone from human GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197425(CHEMBL440227 | [4-({[4-((9S,11R,13S,14S,17S)-17-hy...)
Affinity DataKi:  4.40nMAssay Description:Inhibition of human GR expressed in hGRAF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197425(CHEMBL440227 | [4-({[4-((9S,11R,13S,14S,17S)-17-hy...)
Affinity DataKi:  32nMAssay Description:Inhibition of human GR transcriptional activation by HepTAT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed