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Found 5 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1' and Ligand = 'BDBM50208073'
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(CHEMBL221821 | ginkgolide C)
Affinity DataIC50:  1.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(CHEMBL221821 | ginkgolide C)
Affinity DataIC50:  2.40E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(CHEMBL221821 | ginkgolide C)
Affinity DataIC50:  2.40E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 30 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(CHEMBL221821 | ginkgolide C)
Affinity DataIC50:  4.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50208073(CHEMBL221821 | ginkgolide C)
Affinity DataIC50:  5.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 3000 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed