Found 3 Enz. Inhib. hit(s) with Target = 'Glycine receptor subunit alpha-1' and Ligand = 'BDBM50251276'
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells assessed as inhibition of 300 uM glycine-induced current by whole-cell patch clamp experimentMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Activity at human alpha1betaGlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair
TargetGlycine receptor subunit alpha-1(Homo sapiens (Human))
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 2.90E+3nMAssay Description:Activity at human alpha1GlyR expressed in HEK293 cells by FMP assayMore data for this Ligand-Target Pair