Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM294077'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(1-Benzyl-N′-dodecanoyl-4-hydroxy-2-oxo-1,2-d...)
Affinity DataIC50:  5.51E+3nMT: 2°CAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of kinase-Glo. The recombinant human GSK3 enzyme (catalogue no. 14-306...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(1-Benzyl-N′-dodecanoyl-4-hydroxy-2-oxo-1,2-d...)
Affinity DataIC50:  5.51E+3nMAssay Description:Allosteric inhibition of human recombinant full length N-terminal GST-tagged GSK3beta expressed in fall armyworm Sf9 cells after 30 min in presence o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Consejo Superior de Investigaciones Cientificas (CSIC)

US Patent
LigandPNGBDBM294077(1-Benzyl-N′-dodecanoyl-4-hydroxy-2-oxo-1,2-d...)
Affinity DataIC50:  5.51E+3nMAssay Description:The enzyme inhibition assays were performed using the luminometric methodology of Kinase-GloŽ. The recombinant human GSK3 enzyme (catalogue no. 14-30...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent