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Found 3 Enz. Inhib. hit(s) with Target = 'Glycogen synthase kinase-3 beta' and Ligand = 'BDBM50365609'
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Crystalgenomics

Curated by ChEMBL
LigandPNGBDBM50365609(CHEMBL1957956)
Affinity DataIC50:  3nMAssay Description:Inhibition of GSK3-betaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Crystalgenomics

Curated by ChEMBL
LigandPNGBDBM50365609(CHEMBL1957956)
Affinity DataEC50:  490nMAssay Description:Inhibition of GSK3-beta in human RD cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Crystalgenomics

Curated by ChEMBL
LigandPNGBDBM50365609(CHEMBL1957956)
Affinity DataEC50:  100nMAssay Description:Inhibition of GSK3-beta in human RD cells assessed as glycogen synthase activation measured after 24 hrs under serum starving conditionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed