Found 8 Enz. Inhib. hit(s) with Target = 'Heat shock protein HSP 90-beta' and Ligand = 'BDBM50180302'
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 42nMAssay Description:Displacement of Cy3B-GM from recombinant Hsp90beta (unknown origin) after 24 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of Her2 degradation in human breast cancer SKBr3 cell lineMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataEC50: 6.00E+3nMAssay Description:Binding affinity to Hsp90 in heart tissueMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataEC50: 16.1nMAssay Description:Inhibitory activity against Hsp90 in human breast cancer SKBr3 cell lineMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Inhibition of Hsp90 in human SKBR3 cells assessed as Her2 degradationMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataEC50: 10.2nMAssay Description:Inhibitory activity against Hsp90 in human breast cancer MDA-MB-468 cell lineMore data for this Ligand-Target Pair
TargetHeat shock protein HSP 90-beta(Homo sapiens (Human))
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Sloan-Kettering Institute For Cancer Research
Curated by ChEMBL
Affinity DataEC50: 2.20E+3nMAssay Description:Binding affinity to Hsp90 in lung tissueMore data for this Ligand-Target Pair