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Found 3 Enz. Inhib. hit(s) with Target = 'Hepatocyte growth factor receptor' and Ligand = 'BDBM388836'
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM388836(2-Fluoro-N-(1-pyridin-2-ylcyclopropyl)-4-[3-(1-qui...)
Affinity DataIC50: <500nMAssay Description:Compounds were screened in vitro for their ability to inhibit c-Met kinase activity. The IC50 values of compounds for the inhibition of c-Met kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM388836(2-Fluoro-N-(1-pyridin-2-ylcyclopropyl)-4-[3-(1-qui...)
Affinity DataIC50: <500nMAssay Description:Compounds were screened in vitro for their ability to inhibit c-Met kinase activity. The IC50 values of compounds for the inhibition of c-Met kinase ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHepatocyte growth factor receptor(Homo sapiens (Human))
Incyte

US Patent
LigandPNGBDBM388836(2-Fluoro-N-(1-pyridin-2-ylcyclopropyl)-4-[3-(1-qui...)
Affinity DataIC50: <500nMAssay Description:Briefly, histidine-tagged c-Met catalytic domain fusion protein was used for the assay. IC50 measurements were based on the degree of phosphorylation...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent