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Found 5 Enz. Inhib. hit(s) with Target = 'Histamine H2 receptor' and Ligand = 'BDBM86740'
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  12nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  23nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataKi:  67nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86740(UR-AK24 | UR-AK57)
Affinity DataEC50:  67.6nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig spontaneously beating right atrium assessed as positive chronotropic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed