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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H2 receptor' and Ligand = 'BDBM86743'
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86743(UR-AK49)
Affinity DataKi:  22nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86743(UR-AK49)
Affinity DataKi:  46nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Cavia porcellus (domestic guinea pig))
University Of Kansas

Curated by PDSP Ki Database
LigandPNGBDBM86743(UR-AK49)
Affinity DataEC50:  61.7nMAssay Description:Agonist activity at histamine H2 receptor in guinea pig spontaneously beating right atrium assessed as positive chronotropic activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed