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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50328812'
TargetHistamine H3 receptor(Homo sapiens (Human))
Athersys

Curated by ChEMBL
LigandPNGBDBM50328812(CHEMBL1270264 | rac-1,2,5-trimethyl-4-(quinolin-5-...)
Affinity DataIC50:  12nMAssay Description:Antagonist activity against human histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Mus musculus)
Athersys

Curated by ChEMBL
LigandPNGBDBM50328812(CHEMBL1270264 | rac-1,2,5-trimethyl-4-(quinolin-5-...)
Affinity DataIC50:  690nMAssay Description:Antagonist activity against mouse histamine H3 receptor expressed in human HT1080 cells assessed as inhibition of (R)-alpha-methylhistamine-induced i...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed