Affinity DataKi: 5nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Inverse agonist activity at human histamine H3 histamine receptor by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair