Affinity DataKi: 2.70nMAssay Description:Displacement of [3H]NAMH from human histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D
Curated by ChEMBL
Teva Pharmaceutical Global R & D
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor transfected in CHO cellsMore data for this Ligand-Target Pair
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Teva Pharmaceutical Global R & D
Curated by ChEMBL
Teva Pharmaceutical Global R & D
Curated by ChEMBL
Affinity DataKi: 4.40nMAssay Description:Displacement of [3H]NAMH from rat histamine H3 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 0.800nMAssay Description:Inverse agonist activity at human histamine H3 receptor assessed as inhibition of R-alpha-methylhistamine-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair