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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50408755'
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50408755(CHEMBL2145442)
Affinity DataKi:  9.40nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Freie UniversitäT Berlin

Curated by ChEMBL
LigandPNGBDBM50408755(CHEMBL2145442)
Affinity DataEC50:  0.25nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed