Affinity DataKi: 9.40nMAssay Description:In vitro binding affinity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair
Affinity DataEC50: 0.25nMAssay Description:In vitro intrinsic activity against histamine H3 receptor from synaptosomes of rat cerebral cortexMore data for this Ligand-Target Pair