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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50412461'
TargetHistamine H3 receptor(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50412461(CHEMBL457004)
Affinity DataKi:  0.871nMAssay Description:Displacement of [3H]RAMHA from human histamine H3 receptor expressed in SK-N-MC cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
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Curated by ChEMBL
LigandPNGBDBM50412461(CHEMBL457004)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]RAMHA from histamine H3 receptor in Wistar rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed