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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H4 receptor' and Ligand = 'BDBM294386'
TargetHistamine H4 receptor(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM294386(US9586959, Compound 49)
Affinity DataIC50:  34nMAssay Description:Displacement of [3H]-histamine from recombinant human histamine H4 receptor expressed in CHO-K1 cell membranes measured after 30 mins by microbeta sc...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Sungkyunkwan University

Curated by ChEMBL
LigandPNGBDBM294386(US9586959, Compound 49)
Affinity DataIC50:  34nMpH: 7.5 T: 2°CAssay Description:In vitro profiling protein kinases was performed using the HotSpot assay platform. Briefly, specific kinase/substrate pairs along with required cofac...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent