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Found 2 Enz. Inhib. hit(s) with Target = 'Histone-arginine methyltransferase CARM1' and Ligand = 'BDBM440404'
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Epizyme

US Patent
LigandPNGBDBM440404(US10633389, Example 69-3 | US20230279020, Example ...)
Affinity DataIC50: <100nMAssay Description:The assays were all performed in a buffer consisting of 20 mM Bicine (pH=7.6), 1 mM TCEP, 0.005% BSG, and 0.002% Tween 20, prepared on the day of use...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Epizyme

US Patent
LigandPNGBDBM440404(US10633389, Example 69-3 | US20230279020, Example ...)
Affinity DataIC50: <100nMAssay Description:The assays were all performed in a buffer consisting of 20 mM Bicine (pH=7.6), 1 mM TCEP, 0.005% BSG, and 0.002% Tween 20, prepared on the day of use...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent