Found 5 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase SETD7' and Ligand = 'BDBM50001750' TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Rockefeller University
Curated by ChEMBL
Rockefeller University
Curated by ChEMBL
Affinity DataIC50: 9.93E+3nMAssay Description:Inhibition of methyl-transferase activity in GST-tagged recombinant SET7/9 (unknown origin) expressed in Escherichia coli BL21 using H3(1-20)-cys-bio...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Rockefeller University
Curated by ChEMBL
Rockefeller University
Curated by ChEMBL
Affinity DataIC50: 1.90E+4nMAssay Description:Inhibition of 10 nM SET7 (unknown origin)-mediated methylation of histone H3(1-20)cys-biotin at 15 to 50 uM after 5 mins by scintillation proximity a...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Rockefeller University
Curated by ChEMBL
Rockefeller University
Curated by ChEMBL
Affinity DataIC50: 1.95E+4nMAssay Description:Inhibition of 100 nM SET7 (unknown origin)-mediated methylation of histone H3(1-20)cys-biotin at 15 to 50 uM after 5 mins by scintillation proximity ...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Rockefeller University
Curated by ChEMBL
Rockefeller University
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of 50 nM SET7 (unknown origin)-mediated methylation of histone H3(1-20)cys-biotin at 15 to 50 uM after 5 mins by scintillation proximity a...More data for this Ligand-Target Pair
TargetHistone-lysine N-methyltransferase SETD7(Homo sapiens (Human))
Rockefeller University
Curated by ChEMBL
Rockefeller University
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Inhibition of SET7 (unknown origin)-mediated methylation of histone H3(1-20)cys-biotin after 5 mins by scintillation proximity assay in presence of [...More data for this Ligand-Target Pair
