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Found 3 Enz. Inhib. hit(s) with Target = 'Hydroxycarboxylic acid receptor 2' and Ligand = 'BDBM23532'
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM23532(2-{3-[1-(5-hydroxypyridin-2-yl)-1H-pyrazol-3-yl]pr...)
Affinity DataIC50:  58nM EC50:  1.30E+3nMpH: 7.4 T: 2°CAssay Description:Membranes were incubated in binding buffer with [5, 6-3H]-niacin in the presence of test compound. After 4 hours at room temperature, reactions were ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM23532(2-{3-[1-(5-hydroxypyridin-2-yl)-1H-pyrazol-3-yl]pr...)
Affinity DataIC50:  58nMAssay Description:Displacement of [3H]niacin from GRP109A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM23532(2-{3-[1-(5-hydroxypyridin-2-yl)-1H-pyrazol-3-yl]pr...)
Affinity DataEC50:  1.30E+3nMAssay Description:Displacement of [3H]niacin from GRP109A receptor in presence of 4% human serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed