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Found 2 Enz. Inhib. hit(s) with Target = 'Kappa-type opioid receptor' and Ligand = 'BDBM50010534'
TargetKappa-type opioid receptor(Mus musculus (Mouse))
Eisai

Curated by ChEMBL
LigandPNGBDBM50010534(2-[2-(2-{2-[3-(4-Hydroxy-phenyl)-2-methylamino-pro...)
Affinity DataKi:  1.90nMAssay Description:Binding affinities against Opioid receptor kappa 1 of guinea pig brain membrane using [3H]U69,593 as the radioligand using competition binding assays...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Eisai

Curated by ChEMBL
LigandPNGBDBM50010534(2-[2-(2-{2-[3-(4-Hydroxy-phenyl)-2-methylamino-pro...)
Affinity DataIC50:  2.60nMAssay Description:Evaluated for inhibitory activity against Opioid receptor kappa 1 of rabbit vas deferens (RVD)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed