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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Lysine-specific demethylase 4C (JMJD2C)' and Ligand = 'BDBM340042'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Lysine-specific demethylase 4C (JMJD2C)


(Homo sapiens (Human))
BDBM340042
PNG
(2-(6-Chloro-2-methyl-2H-indazol-3-yl)-1H-pyrrolo[3...)
Show SMILES Cn1nc2cc(Cl)ccc2c1-c1cc2nccc(C(O)=O)c2[nH]1
Show InChI InChI=1S/C16H11ClN4O2/c1-21-15(9-3-2-8(17)6-11(9)20-21)13-7-12-14(19-13)10(16(22)23)4-5-18-12/h2-7,19H,1H3,(H,22,23)
PDB

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/a 550n/an/an/an/an/an/a



CELGENE QUANTICEL RESEARCH, INC.

US Patent


Assay Description
The ability of test compounds to inhibit the activity of JMJD2C was determined in 384-well plate format under the following reaction conditions: 0.3 ...


US Patent US9758517 (2017)

More data for this
Ligand-Target Pair