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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Mast/stem cell growth factor receptor Kit' and Ligand = 'BDBM346158'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Mast/stem cell growth factor receptor Kit


(Homo sapiens (Human))
BDBM346158
PNG
(US10202370, Example 092 | [1-Methyl-2-(3- trifluor...)
Show SMILES Cn1c(nc2cc(Nc3nc(cs3)-c3cccnc3)ccc12)-c1cccc(OC(F)(F)F)c1
Show InChI InChI=1S/C23H16F3N5OS/c1-31-20-8-7-16(28-22-30-19(13-33-22)15-5-3-9-27-12-15)11-18(20)29-21(31)14-4-2-6-17(10-14)32-23(24,25)26/h2-13H,1H3,(H,28,30)
PDB

UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
US Patent
n/an/an/an/a 5.50E+3n/an/an/an/a



AB SCIENCE

US Patent


Assay Description
Colorimetric cell proliferation and viability assay (reagent CellTiter-Blue purchased from Promega cat NG8081) was performed on BaF3 Kit WT cell lin...


US Patent US10202370 (2019)

More data for this
Ligand-Target Pair