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Found 2 Enz. Inhib. hit(s) with Target = 'Melanin-concentrating hormone receptor 1' and Ligand = 'BDBM50168507'
TargetMelanin-concentrating hormone receptor 1(Homo sapiens (Human))
Procter And Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50168507((E)-N-(1-cinnamylpiperidin-4-yl)-3,5-dimethoxybenz...)
Affinity DataKi:  12nMAssay Description:Binding activity against human MCH-R1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanin-concentrating hormone receptor 1(Mus musculus)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50168507((E)-N-(1-cinnamylpiperidin-4-yl)-3,5-dimethoxybenz...)
Affinity DataIC50:  170nMAssay Description:Inhibitory concentration required for binding affinity against mouse MCHr1 competing human neuronal IMR32 cells receptor in a radiometric binding ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed