Affinity DataKi: 140nMAssay Description:Binding affinity against human melanocortin receptor 3 (hMC3R) (concentration of the peptide at 50% specific binding)More data for this Ligand-Target Pair
Affinity DataIC50: 3.30nMAssay Description:Inhibitory activity against human Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataEC50: 2.80nMAssay Description:Evaluated for agonist activity at cloned Melanocortin 3 receptorMore data for this Ligand-Target Pair
Affinity DataKd: 5nMAssay Description:Evaluated for partial agonistic activity at cloned mammalian Melanocortin 3 receptorMore data for this Ligand-Target Pair