TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataKi: 125nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataKi: 736nMAssay Description:Inhibitory activity towards human Melanocortin 3 ReceptorMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Displacement of [125I]NDP-MSH from HEK293 cells expressing human melanocortin-3 receptorMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataIC50: 761nMAssay Description:Displacement of [125I]NDP-alpha-MSH from human MC3R expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataIC50: 761nMAssay Description:Evaluated for binding affinity against human Melanocortin-3 receptor (hMC3R) by displacing [125I]NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataIC50: 761nMAssay Description:Concentration required for 50% inhibition by displacement of of [125I]NDP-alpha-MSH of human MC3R expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.88E+3nMAssay Description:Evaluated for binding affinity against rat Melanocortin-3 receptor (rMC3R) by displacing [125I]-NDP-alpha-MSH radioligand expressed in CHO cellsMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 160nMAssay Description:Agonist activity at human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.33E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in rat Melanocortin-3 receptor (rMC3R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 2.49E+3nMAssay Description:Activity against human MC3R by cAMP accumulationMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 1.40E+3nMAssay Description:In vitro cAMP accumulation in HEK cells transfected with human Melanocortin 3 receptor (hMC3R)More data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 2.49E+3nMAssay Description:Functional activity as concentration of the compound at 50% maximum cAMP accumulation in human melanocortin 1 (MC3R) receptorMore data for this Ligand-Target Pair
TargetMelanocortin receptor 3(Homo sapiens (Human))
Nanyang Technological University
Curated by ChEMBL
Nanyang Technological University
Curated by ChEMBL
Affinity DataEC50: 2.49E+3nMAssay Description:Evaluated for Functional Activity at MC3R as effective concentration at 50% maximum CMP accumulationMore data for this Ligand-Target Pair