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Found 2 Enz. Inhib. hit(s) with Target = 'Melanocortin receptor 4' and Ligand = 'BDBM50182081'
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182081(CHEMBL205461 | N-[2-(5-bromo-2-methoxy-benzyloxy)-...)
Affinity DataKi:  900nMAssay Description:Binding affinity to MC4R by membrane filtration assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
Millennium Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50182081(CHEMBL205461 | N-[2-(5-bromo-2-methoxy-benzyloxy)-...)
Affinity DataIC50:  530nMAssay Description:Antagonist activity against MC4R by cAMP functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed