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Found 4 Enz. Inhib. hit(s) with Target = 'Melanocyte-stimulating hormone receptor' and Ligand = 'BDBM50189020'
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189020(CHEMBL387246 | D-Phe-Arg-2-Nal-NHCH3)
Affinity DataKi:  4.38E+3nMAssay Description:Binding affinity to human MC1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189020(CHEMBL387246 | D-Phe-Arg-2-Nal-NHCH3)
Affinity DataKi:  4.38E+3nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189020(CHEMBL387246 | D-Phe-Arg-2-Nal-NHCH3)
Affinity DataEC50:  2.00E+4nMAssay Description:Displacement of europium labeled NDP-alpha-MSH from human MC1R expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocyte-stimulating hormone receptor(Homo sapiens (Human))
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50189020(CHEMBL387246 | D-Phe-Arg-2-Nal-NHCH3)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human MC1RMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed