BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM361365'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))
BDBM361365
PNG
(3-neopentyl-N- (1H-pyrazolo[3,4- b]pyridin-3-yl)be...)
Show SMILES CC(C)(C)Cc1nsc2cc(Nc3n[nH]c4ncccc34)ccc12
Show InChI InChI=1S/C18H19N5S/c1-18(2,3)10-14-12-7-6-11(9-15(12)24-23-14)20-17-13-5-4-8-19-16(13)21-22-17/h4-9H,10H2,1-3H3,(H2,19,20,21,22)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/an/an/a 884n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...


US Patent US10221172 (2019)


Article DOI: 10.1021/jm070728r
More data for this
Ligand-Target Pair