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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM361372'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))
BDBM361372
PNG
(N-(1H-pyrazolo[3,4-b] pyridin-3-yl)-3- (trifluorom...)
Show SMILES FC(F)(F)c1nsc2cc(Nc3n[nH]c4ncccc34)ccc12
Show InChI InChI=1S/C14H8F3N5S/c15-14(16,17)11-8-4-3-7(6-10(8)23-22-11)19-13-9-2-1-5-18-12(9)20-21-13/h1-6H,(H2,18,19,20,21)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/an/an/a 1.24E+3n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...


US Patent US10221172 (2019)


Article DOI: 10.1021/jm070728r
More data for this
Ligand-Target Pair