BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM361378'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))
BDBM361378
PNG
(3-cyclopropyl-N- (1H-pyrazolo [4,3-b]pyridin-3-yl)...)
Show SMILES C1CC1c1nsc2cc(Nc3n[nH]c4cccnc34)ccc12
Show InChI InChI=1S/C16H13N5S/c1-2-12-15(17-7-1)16(20-19-12)18-10-5-6-11-13(8-10)22-21-14(11)9-3-4-9/h1-2,5-9H,3-4H2,(H2,18,19,20)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/an/an/a 78.2n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...


US Patent US10221172 (2019)


Article DOI: 10.1021/jm070728r
More data for this
Ligand-Target Pair