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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM361382'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))
BDBM361382
PNG
(3-(sec-butyl)-N-(1H- pyrazolo[4,3-b]pyridin- 3-yl)...)
Show SMILES CCC(C)c1nsc2cc(Nc3n[nH]c4cccnc34)cnc12
Show InChI InChI=1/C16H16N6S/c1-3-9(2)13-15-12(23-22-13)7-10(8-18-15)19-16-14-11(20-21-16)5-4-6-17-14/h4-9H,3H2,1-2H3,(H2,19,20,21)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/an/an/a 54.2n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...


US Patent US10221172 (2019)


Article DOI: 10.1021/jm070728r
More data for this
Ligand-Target Pair