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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 4' and Ligand = 'BDBM361390'   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 4


(Homo sapiens (Human))
BDBM361390
PNG
(3-methyl-N-(1H-pyrazolo [3,4-b]pyridin-3- yl)isoth...)
Show SMILES Cc1nsc2cc(Nc3n[nH]c4ncccc34)cnc12
Show InChI InChI=1S/C13H10N6S/c1-7-11-10(20-19-7)5-8(6-15-11)16-13-9-3-2-4-14-12(9)17-18-13/h2-6H,1H3,(H2,14,16,17,18)
UniProtKB/SwissProt

GoogleScholar
PC cid
PC sid
UniChem
Article
US Patent
n/an/an/an/a 180n/an/an/an/a



Vanderbilt University

US Patent


Assay Description
In the first mode, a range of concentrations of the disclosed compounds are added to cells, followed by a single fixed concentration of agonist. If t...


US Patent US10221172 (2019)


Article DOI: 10.1021/jm070728r
More data for this
Ligand-Target Pair