Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase 1' and Ligand = 'BDBM203364'
Affinity DataIC50: 3nMAssay Description:Activated ERK2 activity was also determined in the IMAP assay format using the procedure outlined above. 1 μl of 25× compound was added to 14 ...More data for this Ligand-Target Pair
Affinity DataKd: 0.140nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by
this invention was interrogated using the TdF (Temperature Dependence
Fluoresc...More data for this Ligand-Target Pair