Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 12' and Ligand = 'BDBM365232'
TargetMitogen-activated protein kinase kinase kinase 12(Homo sapiens (Human))
Genentech

US Patent
LigandPNGBDBM365232((2-Pyrrolidin-1-yl-6-pyr- rolidin-3-yl-pyrimidin- ...)
Affinity DataKi:  4.80nMAssay Description:DLK kinase reactions (20 μL) containing 5 nM N-terminally GST-tagged DLK (catalytic domain amino acid 1-520) (Carna Bioscience), 40 nM N-termina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent