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Found 2 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 5' and Ligand = 'BDBM307615'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Seal Rock Therapeutics

US Patent
LigandPNGBDBM307615(2-(6-(4-cyclopropyl- 4H-1,2,4-triazol-3- yl)pyridi...)
Affinity DataKi: <200nMAssay Description:The ASK1 enzymatic assay was run following Promega ASK1 Kinase Enzyme System (Cat #V3881). The kit provides the protocol, enzymes and all reagents ne...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Seal Rock Therapeutics

US Patent
LigandPNGBDBM307615(2-(6-(4-cyclopropyl- 4H-1,2,4-triazol-3- yl)pyridi...)
Affinity DataIC50: <200nMAssay Description:The ASK1 enzymatic assay was run following Promega ASK1 Kinase Enzyme System (Cat #V3881). The kit provides the protocol, enzymes and all reagents ne...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent