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Found 1 Enz. Inhib. hit(s) with Target = 'Mitogen-activated protein kinase kinase kinase 5' and Ligand = 'BDBM419023'
TargetMitogen-activated protein kinase kinase kinase 5(Homo sapiens (Human))
Enanta Pharmaceuticals

US Patent
LigandPNGBDBM419023(US10450301, Example 102)
Affinity DataIC50:  55nMAssay Description:HTRF KinEASE-STK is a generic method for measuring serine/threonine kinase activities using a time-resolved fluorescence resonance energy transfer (T...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent