Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Monoglyceride lipase' and Ligand = 'BDBM50255235'
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50255235(CHEMBL4078924)
Affinity DataKi:  412nMAssay Description:Competitive inhibition of recombinant human MAGL using 4-NPA as substrate after 30 mins by Michaelis-Menten plot analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50255235(CHEMBL4078924)
Affinity DataIC50:  390nMAssay Description:Inhibition of recombinant human MAGL using 4-NPA as substrate after 30 mins by colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50255235(CHEMBL4078924)
Affinity DataIC50:  500nMAssay Description:Inhibition of recombinant human MAGL using 4-NPA as substrate after 10 mins in presence of DTT by colorimetric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50255235(CHEMBL4078924)
Affinity DataIC50:  510nMAssay Description:Inhibition of recombinant human MAGL using 4-NPA as substrate after 10 mins by HPLC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed