Affinity DataKi: 2.20nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 5.51nMAssay Description:Inhibition of binding of [3H]naloxone to Opioid receptor mu 1 in the rat brain homogenateMore data for this Ligand-Target Pair
Affinity DataIC50: 7.60nMAssay Description:Inhibitory potency against mu receptor in guinea pig ileum assayMore data for this Ligand-Target Pair