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Found 2 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM50174852'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174852(CHEMBL198648 | rac-N-((3-(9-chloro-3-methyl-4-oxoi...)
Affinity DataIC50:  270nMAssay Description:Inhibitory activity against MRP1-mediated LTC4 uptake into membrane vesicles from HeLa-T5 cells expressing MRP1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50174852(CHEMBL198648 | rac-N-((3-(9-chloro-3-methyl-4-oxoi...)
Affinity DataEC50:  250nMAssay Description:Inhibitory activity against MRP1 in HeLa-T5 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed