Found 4 Enz. Inhib. hit(s) with Target = 'Multidrug resistance-associated protein 1' and Ligand = 'BDBM67690'
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-M24 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-M6 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:TP_TRANSPORTER: cell accumulation in MCF7/MRP1-10 cellsMore data for this Ligand-Target Pair
TargetMultidrug resistance-associated protein 1(Homo sapiens (Human))
Wake Forest University School Of Medicine
Curated by ChEMBL
Wake Forest University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of MRP1 in human 2008/MRP1 cells assessed as reduction in cell viability after 5 days by MTS/PMS assayMore data for this Ligand-Target Pair