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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM261732'
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM261732(1-fluoro-N- ((3RS,4SR)-3- hydroxytetrahydro- 2H-py...)
Affinity DataEC50:  3nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent
LigandPNGBDBM261732(1-fluoro-N- ((3RS,4SR)-3- hydroxytetrahydro- 2H-py...)
Affinity DataEC50:  2nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent
LigandPNGBDBM261732(1-fluoro-N- ((3RS,4SR)-3- hydroxytetrahydro- 2H-py...)
Affinity DataEC50:  6nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM261732(1-fluoro-N- ((3RS,4SR)-3- hydroxytetrahydro- 2H-py...)
Affinity DataEC50:  2nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent