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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Ligand = 'BDBM261740'
TargetMuscarinic acetylcholine receptor M1(RAT)
Hoffmann-La Roche

US Patent
LigandPNGBDBM261740(4-((4-Cyano-4-(pyridin-2-yl)piperidin-1-yl)methyl)...)
Affinity DataEC50:  345nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Hoffmann-La Roche

US Patent
LigandPNGBDBM261740(4-((4-Cyano-4-(pyridin-2-yl)piperidin-1-yl)methyl)...)
Affinity DataEC50:  258nMAssay Description:The assay is designed to select compounds that possess modulator activity at the acetylcholine muscarinic receptor expressed in CHO cells by measurin...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent