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Found 4 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Ligand = 'BDBM50004737'
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50004737(3-Methyl-1-(4-pyrrolidin-1-yl-but-2-ynyl)-pyrrolid...)
Affinity DataKi:  15nMAssay Description:Binding affinity at [3H]CD radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50004737(3-Methyl-1-(4-pyrrolidin-1-yl-but-2-ynyl)-pyrrolid...)
Affinity DataKi:  80nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50004737(3-Methyl-1-(4-pyrrolidin-1-yl-but-2-ynyl)-pyrrolid...)
Affinity DataKi:  710nMAssay Description:Binding affinity at [3H]QNB radiolabeled muscarinic M2 receptor in rat cortex.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M2(RAT)
Medical Research Division Of American Cyanamid

Curated by ChEMBL
LigandPNGBDBM50004737(3-Methyl-1-(4-pyrrolidin-1-yl-but-2-ynyl)-pyrrolid...)
Affinity DataKi:  1.10E+3nMAssay Description:Binding affinity at [3H]QNB and GppNHp radiolabeled muscarinic M2 receptor in rat heart.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed